The first direct chemical inhibitor of a key histone-methylating enzyme provides a new tool to alter epigenetic states and genome expression profiles in normal and cancer cells.
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Simon, J. Stopping a chromatin enzyme. Nat Chem Biol 8, 875–876 (2012). https://doi.org/10.1038/nchembio.1088
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DOI: https://doi.org/10.1038/nchembio.1088