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This work was supported by National Natural Science Foundation of China (#81573277, 81622042, and 81773567), National Major Scientific and Technological Special Project for “Significant New Drugs Development” (#SQ2017ZX095003), and Tsinghua University Initiative Scientific Research Program. This work was also financially supported by NSFC (No. 81670187) and Beijing Natural Science Foundation (No. 7172047).
Conflict of interest
The authors declare that they have no conflict of interest.
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Sun, Y., Ding, N., Song, Y. et al. Degradation of Bruton’s tyrosine kinase mutants by PROTACs for potential treatment of ibrutinib-resistant non-Hodgkin lymphomas. Leukemia 33, 2105–2110 (2019) doi:10.1038/s41375-019-0440-x
Future Medicinal Chemistry (2019)