Degradation of Bruton’s tyrosine kinase mutants by PROTACs for potential treatment of ibrutinib-resistant non-Hodgkin lymphomas

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This work was supported by National Natural Science Foundation of China (#81573277, 81622042, and 81773567), National Major Scientific and Technological Special Project for “Significant New Drugs Development” (#SQ2017ZX095003), and Tsinghua University Initiative Scientific Research Program. This work was also financially supported by NSFC (No. 81670187) and Beijing Natural Science Foundation (No. 7172047).

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Correspondence to Wanli Liu or Jun Zhu or Yu Rao.

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Sun, Y., Ding, N., Song, Y. et al. Degradation of Bruton’s tyrosine kinase mutants by PROTACs for potential treatment of ibrutinib-resistant non-Hodgkin lymphomas. Leukemia 33, 2105–2110 (2019) doi:10.1038/s41375-019-0440-x

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