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Interrogating the kinome

Comprehensive studies of the kinome set the stage for discovering the next generation of kinase-directed drugs.

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Figure 1: Kinome-wide investigation of kinase inhibitor selectivity.

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Correspondence to Gideon Bollag.

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The authors are employees of Plexxikon Inc., a member of the Daiichi Sankyo group.

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Zhang, C., Habets, G. & Bollag, G. Interrogating the kinome. Nat Biotechnol 29, 981–983 (2011). https://doi.org/10.1038/nbt.2021

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