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Nature Structural & Molecular Biology 11, 1192–1197 (1 December 2004) | doi:10.1038/nsmb859

Structures of human MAP kinase kinase 1 (MEK1) and MEK2 describe novel noncompetitive kinase inhibition

Jeffrey F Ohren , Huifen Chen , Alexander Pavlovsky , Christopher Whitehead , Erli Zhang , Peter Kuffa , Chunhong Yan , Patrick McConnell , Cindy Spessard , Craig Banotai , W Thomas Mueller , Amy Delaney , Charles Omer , Judith Sebolt-Leopold , David T Dudley , Iris K Leung , Cathlin Flamme , Joseph Warmus , Michael Kaufman , Stephen Barrett , Haile Tecle & Charles A Hasemann