Table 1


From the following article

Antivirals—an increasingly healthy investment

Brian McCarthy

Nature Biotechnology 25, 1390 - 1393 (2007)

doi:10.1038/nbt1207-1390

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Table 1. HIV therapeutics with recent or imminent patent expirations

CompanyDrug (generic name)PatentDate of expiration
 Nucleoside analog reverse transcriptase inhibitor
Bristol-Myers SquibbVidex (dideoxyinosine)US 5,254,539March 2007
Bristol-Myers SquibbZerit (stavudine; d4T)VariousJune 2008
Glaxo WellcomeZiagen (abacavir)VariousJune–December 2009
Glaxo WellcomeCombivir (lamivudine/zidovudine)US 5,859,021May 2012
GileadEmtriva (emtricitabine)US 5,210,085July 2008
Hoffmann-La RocheZalcitabine (ddC)VariousJuly 2008
 Protease inhibitor
Hoffmann-La RocheInvirase/Fortovase (saquinavir mesylate)US 5,196,438November 2010
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