Kidney International (1994) 45, 692–699; doi:10.1038/ki.1994.93
Effects of neurohypophyseal antagonists in postnephrectomy natriuresis in male rats
Wan Huang1, Siu-Lan Lee1 and Mats Sjöquist1
1Department of Physiology and Medical Biophysics, Biomedicum, Uppsala University, Uppsala, Sweden
Correspondence: Mats Sjöquist, Departments of Physiology and Medical Biophysics, Biomedicum, Uppsala University, Box 572, S-751 23 Uppsala, Sweden.
Received 13 October 1992; Revised 20 September 1993; Accepted 20 September 1993.
Top of pageAbstract
Effects of neurohypophyseal antagonists in postnephrectomy natriuresis in male rats. Acute unilateral nephrectomy (AUN) in anesthetized male Lewis x DA rats induced rapid and consistent increases in electrolyte and fluid excretion by the remaining kidney during the first hours. Continuous infusion of a vasopressin (AVP) V1-receptor antagonist d(CH2)5 Tyr(Me)AVP (V1-ant) reduced renal electrolyte and fluid excretion before and after AUN to a similar extent, whereas an oxytocin (OT)-receptor antagonist [Mpa1,D-Tyr(Et)2,Thr4,Orn8]-OT (CAP) at the same dose selectively attenuated the increase in sodium excretion after AUN. The plasma concentration of OT rose significantly after AUN (9.16
1.4 to 21.45
5.07 pg
ml-1). A similar OT level obtained by infusion of OT mimicked the renal responses to AUN without elevating blood pressure; however, only CAP but not V1-ant efficiently reversed OT-induced natriuresis. Also, the infusion of CAP at the same dose produced no effects on the rise of blood pressure caused by AVP while the infusion of the V1-ant prevented such a rise. Thus, CAP reduced the natriuresis after AUN by interfering with OT-and not V1-receptors. In conclusion, evidence is presented, for the first time, concerning the major role of OT receptors in the acute readjustment of the renal sodium excretion after AUN, and a synergistic role for AVP in terms of the general magnitude of renal excretion.
Top of pageReferences
- Humphreys MH, Lin S-Y, Wiedemann E: Renal nerves and the natriuresis following unilateral renal exclusion in the rat. Kidney Int 39:63–70, 1991
- Calaresu FR, Ciriello J: Renal afferent nerves affect discharge rate of medullary and hypothalamic single units in the cat. J Auton Nerv Syst 3:311–320, 1981 | Article | PubMed | ISI | ChemPort |
- Lin S-Y, Wiedemann E, Humphreys MH: Role of the pituitary in reflex natriuresis following acute unilateral nephrectomy. Am J Physiol 249:F282–F290, 1985
- Lin S-Y, Chaves C, Windemann E, Humphreys MH: A
-melanocyte stimulating hormone-like peptide causes reflex natriuresis after acute unilateral nephrectomy. Hypertension 10:619–627, 1987 | PubMed | - Valentin J-P, Ribstein J, Pussard E, Mimran A: Role of atrial peptide in the acute natriuretic response to uninephrectomy. Am J Physiol 258:F1054–F1060, 1990
- Kasting NW: Simultaneous and independent release of vasopressin and oxytocin in the rat. Can J Physiol Pharmacol 66:22–26, 1988 | PubMed |
- Balment RJ, Brimble MJ, Forsling ML: Release of oxytocin induced by salt loading and its influence in renal excretion in the male rat. J Physiol (London) 308:439–449, 1980
- Brimble MJ, Balment RJ, Smith CP, Windle RJ, Forsling ML: Influence of oxytocin on sodium excretion in the anaesthetized Brattleboro rat. J Endocrinol 129:49–54, 1991
- Balment RJ, Brimble MJ, Forsling ML, Musabayane CT: The influence of neurohypophysial hormones on renal function on the acutely hypophysectomized rat. J Physiol (London) 381:439–452, 1986
- Balment RJ, Brimble MJ, Forsling ML, Kelly LP, Musabayane CT: A synergistic effect of oxytocin and vasopressin on sodium excretion in the neurohypophysectomized rat. J Physiol (London) 381:453–464, 1986
- Brooks FP, Pickford M: The effect of posterior pituitary hormones on the excretion of electrolytes, in dogs. J Physiol (London) 142:468–493, 1958 | PubMed | ISI | ChemPort |
- Conrad KP, Gellai M, North WG, Valtin H: Influence of oxytocin on renal hemodynamics and electrolyte and water excretion. Am J Physiol 251:F290–F296, 1986
- Forsling ML, Brimble MJ: The role of oxytocin in salt and water balance, in Oxytocin: Clinical and Laboratory Studies, edited by Amico JA, AG Robinson, Oxford, Elsevier Science Publishers BV, 1985, pp. 167–175
- Leng G, Dyball REJ, Russell JA: Neurophysiology of body fluid homeostasis. Comp Biochem Physiol 90A(4):781–788, 1988
- Lote CJ, Thewles A, Wood JA: Vasopressin-induced natriuresis in the conscious rat: Role of blood pressure, renal prostaglandin synthesis and the peptide ANF. J Physiol (London) 411:481–491, 1989
- Ulfendahl HR, Ahlsson A, Hansell P, Höglund U, Jacobsson E, Lee SL, Sjöquist M: Studies on the mechanisms underlying CNS-induced natriuresis. Acta Physiol Scand 136(Suppl 583):75–78, 1989
- Lote CJ, Thewles A, Wood JA: Changes in plasma natriuretic factor (ANF), blood pressure and urinary prostaglandin E2 during vasopressin-induced natriuresis in the rat. Pflügers Arch 411(Suppl 1):R88, 1988
- Ayus JC, Humphreys MH: Hemodynamic and renal functional changes after acute unilateral nephrectomy in the dog: Role of carotid sinus baroreceptors. Am J Physiol 242:F181–F189, 1982
- Diezi J, Michoud-Hausel P, Nicolas-Buxcel N: Studies on possible mechanisms of early functional compensatory adaptation in the remaining kidney. Yale J Biol Med 51:265–270, 1978
- Peters G: Compensatory adaptation of renal functions in the unanesthetized rat. Am J Physiol 205(5):1042–1048, 1963
- Johnson MD, Kinter LB, Beeuwkes R III: Effects of AVP and DDAVP on plasma renin activity and electrolyte secretion in conscious dogs. Am J Physiol 236:F66–F70, 1979
- Chan WY, Hruby VJ: Natriuretic action of neurohypophysial peptides: Effects of agonists and antagonists and implication of natriuretic receptor. J Pharmacol Exp Ther 246:597–602, 1988
- Manning M, Sawyer WH: Synthesis and receptor specificities of vasopressin antagonists. J Cardiovasc Pharmacol 8(Suppl 7):S29–S35, 1986
- Melin P: Oxytocin antagonists in preterm labour and delivery. Bailliere's Clin Obstet Gynaecol 7(3):577–600, 1993
- Manning M, Sawyer WH: Design and uses of selective agonistic and antagonistic analogs of the neuropeptides oxytocin and vasopressin. Trends Neurosci 7:6–9, 1984 | ISI | ChemPort |
- Verbalis JG, Mangione MP, Stricker EM: Oxytocin produces natriuresis in rats at physiological plasma concentrations. Endocrinology 128(3):1317–1322, 1991
- Shirley DG, Skinner J: Acute compensatory adaptation of renal function following contralateral kidney exclusion in Brattleboro rats with diabetes insipidus. J Physiol (London) 283:425–438, 1978
- Ribstein J, Humphreys MH: Endogenous opioids and electrolyte excretion after contralateral renal exclusion. Am J Physiol 244:F392–F398, 1983
- Stricker EM, Verbalis JG: Interaction of osmotic and volume stimuli in regulation of neurohypophyseal secretion in rats. Am J Physiol 250:R267–R275, 1986 | PubMed | ChemPort |
- Stoeckel ME, Freund-Mercier MJ: Autoradiographic demonstration of oxytocin-binding sites in the macula densa. Am J Physiol 257:F310–F314, 1989
- Schmidt A, Jard S, Dreifuss JJ, Tribollet E: Oxytocin receptors in rat kidney during development. Am J Physiol 259:F872–F881, 1990 | PubMed |
- Kruszynski M, Lammek B, Manning M, Seto J, Haldar J, Sawyer WH: (1-(B-Mercapto-B,B-cyclopentamethylenepropionic acid),2-(O-methyl)tyrosine)arginine-vasopressin and (1-(B-Mercapto-B,B-cyclopentamehylenepropionic acid))arginine-vasopressin, two highly potent antagonists of the vasopressor response to arginine-vasopressin. J Med Chem 23:364–368, 1980 | Article | PubMed | ISI | ChemPort |