Journal of Investigative Dermatology Symposium Proceedings

TABLE 2

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Latest Insights into Skin Hyperpigmentation

Jean-Paul Ortonne and Donald L Bissett

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Table 2. Pigmentation control targets and effective agents

Pigmentation control target Effective agent
Tyrosinase inhibitionHydroquinone, resorcinols, kojic acid, arbutin, ascorbic acid (vitamin C), deoxyarbutin
Tyrosinase copper chelationEllagic acid
Inhibition of tyrosinase glycosylationGlucosamine, N-acetyl glucosamine, tunicamycin
Melanosome transferNiacinamide, protease inhibitors
Downregulation of tyrosinaseRetinoid (trans-retinoic acid, retinol and its esters, retinaldehyde)
AntioxidantVitamin C compounds, vitamin E, sulfhydryl compounds
Anti-inflammatory agentHydrocortisone, phytosterol, glycyrrhetinic acid
Increase epidermal turnoverRetinoids, salicylic acid
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