7TM Receptors
Subject Category: 7TM Receptors
Citation Information:
We recommend that any citations to information in the Guide are presented
in the following format:
Alexander SPH, Mathie A, Peters JA (2008). Guide to Receptors and Channels (GRAC), 3rd edn. Br J Pharmacol153 (Suppl. 2): S1–S209.
Cannabinoid
S P H Alexander, A Mathie and J A Peters
Keywords:
cannabinoid, anandamide, N-homo-
-linolenylethanolamine, N-docosatetra-7,10,13,16-enylethanolamine, [3H]-CP55940, [3H]-WIN55212-2, ACEA, ACPA, methanandamide, O1812, HU308, JWH133, L759633, L759656, AM1241, AM251, AM281, SR141716A, LY320135, SR144528, AM630, [3H]-SR141716A, vanilloid receptor, GPR55, rimonabant, N-arachidonoylglycine, GPR18, GPR119, N-oleoylethanolamine, N-palmitoylethanolamine, PSN632408, PSN375963
Abbreviations:
ACEA, arachidonoyl-2-chloroethylamide; ACPA, arachidonoylcyclopropylamide; AM1241, (2-iodo-5-nitro-phenyl)-[1-(1-methyl-piperidin-2-ylmethyl)-1H-indol-3-yl]-methanone; AM251, N-(piperidin-1-yl)-5-(4-iodophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-carboxamide; AM281, 1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-4-morpholinyl-1H-pyrazole-3-carboxamide; AM630, 6-iodopravadoline; CP55940, (1R,3R,4R)-3-[2-hydroxy-4-(1,1-dimethylheptyl) phenyl]-4-(3-hydroxypropyl)cyclohexan-1-ol; HU308, {4-[4-(1,1-dimethylheptyl)-2,6-dimethoxy-phenyl]-6,6-dimethyl-bicyclo[3.1.1]hept-2-en-2-yl}-methanol; JWH133, (3-(1,1-dimethylbutyl)-6,6,9-trimethyl-6a,7,10,10a-tetrahydro-6H-benzo[c]chromene; L759633, (6ar,10ar)-3-(1,1-dimethylheptyl)-1-methoxy-6,6,9-trimethyl-6a,7,10,10a-tetrahydro-6H-benzo[c]chromene; L759656, (6ar,10ar)-3-(1,1-dimethylheptyl)-1-methoxy-6,6-dimethyl-9-methylene-6a,7,8,9,10,10a-hexahydro-6H-benzo[c]chromene; LY320135, (6-methoxy-2-[4-methoxyphenyl]benzo[b]thien-3-yl)(4-cyanophenyl)methanone; methanandamide, (R)-(+)-arachidonoyl-1'-hydroxy-2'-propylamide; O1812, (R)-(20-cyano-16,16-dimethyldocosa-cis-5,8,11,14-tetraenoyl)-1'-hydroxy-2'-propylamine; PSN375963, 4-(5-[4-butylcyclohexyl]-1,2,4-oxadiazol-3-yl)pyridine; PSN632408, 4-([3-{4-pyridinyl}-1,2,4-oxadiazol-5-yl]methoxy)-1-piperidinecarboxylic acid, 1,1-dimethylethyl ester; rimonabant, N-(piperidin-1-yl)-5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-carboxamide hydrochloride, also known as SR141716A; SR144528, N-([1S]-endo-1,3,3-trimethylbicyclo[2.2.1]heptan-2-yl)-5-(4-chloro-3-methylphenyl)-1-(4-methylbenzyl)-pyrazole-3-carboxamide; WIN55212-2, (R)-(+)-[2,3-dihydro-5-methyl-3-(4-morpholinylmethyl)pyrrolo-[1,2,3-de]-1,4-benzoxazin-6-yl]-1-naphthalenylmethanone mesylate
